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Supplemental Table 2. TET. HTCA ASSAY. COMPOUND. CLASS. EL. T1. T2. OFF ON. 0.07 μ M ± 0.03 0.05 μ M ± 0.004 0.057 μ M ± 0.01. BJFL018. Meriolins. 0.08 μ M ± 0.02 0.05 μ M ± 0.004 0.058 μ M ± 0.003.
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Supplemental Table 2 TET HTCA ASSAY COMPOUND CLASS EL T1 T2 OFF ON 0.07μM ± 0.03 0.05μM ± 0.004 0.057μM ± 0.01 BJFL018 Meriolins 0.08μM ± 0.02 0.05μM ± 0.004 0.058μM ± 0.003 0.05μM ± 0.01 0.03μM ± 0.004 0.042μM ± 0.02 OFF ON BJFL034 0.05μM ± 0.01 0.031μM ± 0.002 0.041μM ± 0.02 0.26μM ± 0.03 0.75μM ± 0.01 0.27μM ± 0.04 OFF ON C&R-5 0.29μM ± 0.04 0.68μM ± 0.02 0.26μM ± 0.03 0.57μM ± 0.26 1.46μM ± 0.03 0.41μM ± 0.05 OFF ON C&R-6 0.57μM ± 0.22 1.38μM ± 0.08 0.42μM ± 0.02 0.76μM ± 0.07 2.43μM ± 1.04 0.72μM ± 0.05 OFF ON CHOR2 Purines 0.75μM ± 0.05 2.17μM ± 0.83 0.69μM ± 0.04 0.54μM ± 0.18 1.35μM ± 0.07 0.58μM ± 0.04 OFF ON CHOR3 0.57μM ± 0.13 1.35μM ± 0.07 0.57μM ± 0.04 1.43μM ± 0.79 1.08μM ± 0.06 1.34μM ± 0.39 OFF ON CS36 1.46μM ± 0.87 1.02μM ± 0.03 1.23μM ± 0.53 OFF ON 6.67μM ± nd nd 5.13μM ± nd DRF039 7.18μM ± nd nd 5.64μM ± nd